Olodaterol hydrochloride
CAS No. 869477-96-3
Olodaterol hydrochloride ( BI1744 CL )
Catalog No. M16316 CAS No. 869477-96-3
Olodaterol hydrochloride (BI1744 CL) is a potent, selective long-acting β2 adrenoceptor agonist with EC50 of 1.4 nM for hβ2.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
2MG | 71 | In Stock |
|
5MG | 110 | In Stock |
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10MG | 178 | In Stock |
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25MG | 332 | In Stock |
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50MG | 494 | In Stock |
|
100MG | 709 | In Stock |
|
200MG | Get Quote | In Stock |
|
500MG | Get Quote | In Stock |
|
1G | Get Quote | In Stock |
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Biological Information
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Product NameOlodaterol hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionOlodaterol hydrochloride (BI1744 CL) is a potent, selective long-acting β2 adrenoceptor agonist with EC50 of 1.4 nM for hβ2.
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DescriptionOlodaterol hydrochloride (BI1744 CL) is a potent, selective long-acting β2 adrenoceptor agonist with EC50 of 1.4 nM for hβ2; shows >250 fold selectivity over hβ1; exerts a bronchodilatory efficacy over 24 h in dogs and guinea pigs in the absence of systemic pharmacodynamic effects.COPD Phase 3 Clinical
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SynonymsBI1744 CL
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PathwayAngiogenesis
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TargetAdrenergic Receptor
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Recptorhβ2-adrenoceptor
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Research AreaInflammation/Immunology
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IndicationCOPD
Chemical Information
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CAS Number869477-96-3
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Formula Weight413.90
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Molecular FormulaC21H17ClFN3OS
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Purity>98% (HPLC)
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SolubilityDMSO: 50 mg/mL; Water: 15 mg/mL ( < 1 mg/ml refers to the product slightly soluble or insoluble )
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SMILESCC(C)(CC1=CC=C(C=C1)OC)NCC(C2=C3C(=CC(=C2)O)NC(=O)CO3)O.Cl
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Chemical Name4-(4-(4-fluorophenyl)-2-(4-(methylsulfinyl)phenyl)-1H-imidazol-5-yl)pyridine hydrochloride
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Bouyssou T, et al. Bioorg Med Chem Lett. 2010 Feb 15;20(4):1410-4.
2. Bouyssou T, et al. J Pharmacol Exp Ther. 2010 Jul;334(1):53-62.
3. Wex E, et al. Br J Pharmacol. 2015 Jul;172(14):3537-47.
2. Bouyssou T, et al. J Pharmacol Exp Ther. 2010 Jul;334(1):53-62.
3. Wex E, et al. Br J Pharmacol. 2015 Jul;172(14):3537-47.
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